Inhibition of selectin binding by colloidal gold with functionalized shells.

نویسندگان

  • Jens Dernedde
  • Sven Enders
  • Hans-Ulrich Reissig
  • Meike Roskamp
  • Sabine Schlecht
  • Shahla Yekta
چکیده

Gold colloids with terminally functionalized sulfated thiol shells were found to bind to P- and L-selectins with IC(50) values in the picomolar range; branched acyclic epitopes show the highest affinity, whereas a sulfated carbohydrate mimetic provides the best selectivity.

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عنوان ژورنال:
  • Chemical communications

دوره 8  شماره 

صفحات  -

تاریخ انتشار 2009